Byetta vs Rybelsus

exenatide (GLP-1 receptor agonist) vs semaglutide (GLP-1 receptor agonist) — a complete side-by-side comparison.

AstraZenecaNovo Nordisk

Byetta weight loss

2.8%

Rybelsus weight loss

4.4%

Byetta dosing

Twice daily (within 60 min before meals)

Rybelsus dosing

Once daily

Reviewed by Dr. Elena Vance, DOLast reviewed 4 sources cited

Quick Summary

Byetta (exenatide) and Rybelsus (semaglutide) are both glp-1 receptor agonists. In clinical trials, Rybelsus showed greater weight loss (4.4% vs 2.8%).

See the comparison table below for detailed side-by-side data.

Byetta vs Rybelsus: Full Comparison

FeatureByetta(exenatide)Rybelsus(semaglutide)
Active Ingredientexenatidesemaglutide
Drug ClassGLP-1 receptor agonistGLP-1 receptor agonist
ManufacturerAstraZenecaNovo Nordisk
FDA Approved2005-04-282019-09-20
Approved Indications
  • Type 2 diabetes mellitus (adjunct to diet and exercise)
  • Type 2 diabetes mellitus (adjunct to diet and exercise)
Routesubcutaneous injectionoral
FrequencyTwice daily (within 60 min before meals)Once daily
Starting Dose5 mcg twice daily3 mg daily
Maintenance Dose10 mcg twice daily7 mg or 14 mg daily
Max Dose10 mcg twice daily14 mg daily
Weight Loss (%)2.8%4.4%
A1C Reduction0.8%1.4%
Key TrialAC2993 Phase 3 (30 weeks)PIONEER 1 (26 weeks)
List Price$800-$900/month$935-$1,029/month
With Insurance$25-$100/month (varies by plan)$25-$150/month (varies by plan)
Savings CardLimited savings programs available$10/month (Novo Nordisk savings card, commercially insured)

Side Effects: Byetta vs Rybelsus

Side EffectByettaRybelsus
Nausea44%11-20%
Vomiting13%4-8%
Diarrhea13%5-10%
Headache9%Not reported
Dizziness9%Not reported
Dyspepsia6%Not reported
Jittery feeling4%Not reported
Pancreatitis (rare)<1%<0.5%
Abdominal painNot reported5-11%
Decreased appetiteNot reported3-9%
ConstipationNot reported3-5%

Severity scale: 1 (mild) to 5 (serious). Based on FDA prescribing information and clinical trial data.

Related Comparisons

Frequently Asked Questions

Sources & References

  1. Byetta FDA prescribing information
  2. Rybelsus FDA prescribing information
  3. DeFronzo RA et al., Diabetes Care 2005;28:1092-1100.
  4. Aroda VR et al., Lancet 2019;394:39-50. FDA prescribing information.

This content is for informational purposes only and is not medical advice. Always consult your healthcare provider before making medication decisions. See our full medical disclaimer.